Drug Name:
LEVATOL Rx

Generic Name and Formulations:
Penbutolol sulfate 20mg; scored tabs.
Company:
Auxilium Pharmaceuticals, Inc.
Therapeutic Use:
Indications for LEVATOL:
Hypertension.
Adult:
20mg once daily.
Children:
Not recommended.
Contraindications:
Asthma. Cardiogenic shock. Sinus bradycardia. 2nd- or 3rd-degree AV block.
Warnings/Precautions:
Overt heart failure. CHF. Bronchospasm, COPD. Diabetes. Hyperthyroidism. Surgery. Avoid abrupt cessation. Pregnancy (Cat.C). Nursing mothers.
Interactions:
Bradycardia with catecholamine-depleting drugs. May increase cardiac effects of calcium channel blockers, digitalis. Adjust antidiabetic medication. Higher lidocaine loading dose may be needed. May block epinephrine.
Pharmacological Class:
Noncardioselective beta-blocker.
Adverse Reactions:
Bradycardia, headache, dizziness, fatigue, GI upset, cough, dyspnea, insomnia, asthenia, hyperhidrosis, impotence, cardiac failure.
How Supplied:
Tabs—100
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